SCHEMBL19675103

SCHEMBL19675103

COCCCn1nc(C(=O)OF)c2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 8/20 0.47
CNR2 P34972 6/20 0.47
HTR3A P46098 4/20 0.47
HTR4 Q13639 4/20 0.45
REN P00797 1/20 0.43
CYP3A4 P08684 1/20 0.42
F2 P00734 1/20 0.42
PLAU P00749 1/20 0.42
ELANE P08246 1/20 0.42
ALDH1A1 P00352 1/20 0.42
PARP1 P09874 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3071892 0.90 ELANE (0.53) CNR1CNR2HTR3AHTR4CYP3A4
SCHEMBL17324730 0.88 CNR1 (0.48) CNR1CNR2HTR3AHTR4REN
SCHEMBL2808445 0.88 ELANE (0.49) CNR1CNR2HTR3AF2PLAU
SCHEMBL15882396 0.86 ELANE (0.58) CNR1CNR2F2PLAUELANE
SCHEMBL15882017 0.86 CNR1 (0.50) CNR1CNR2CYP3A4
SCHEMBL20250798 0.84 CNR1 (0.49) CNR1CNR2HTR3AHTR4REN
SCHEMBL17321441 0.82 CNR1 (0.51) CNR1CNR2HTR3AHTR4REN
SCHEMBL31429292 0.82 ELANE (0.56) CNR1CNR2HTR3AF2PLAU
SCHEMBL17324818 0.80 KDM4C (0.50) CNR1CNR2HTR3AELANEALDH1A1
SCHEMBL27795771 0.79 ELANE (0.44) CNR1CNR2HTR3AF2PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3252050-A1 PHTHALAZINONES AND ISOQUINOLINONES AS ROCK INHIBITORS Bristol-Myers Squibb Company (US) 2017-12-06 EP disclosed