SCHEMBL19684407

SCHEMBL19684407

CCC(CCN(C)C)NC(=O)c1c(-c2ccnn2-c2ccc(C#N)cc2)n(C)n(-c2cccc(C(F)(F)F)c2)c1=O

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ELANE P08246 15/20 0.49
CTSK P43235 4/20 0.40
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19656241 0.90 ELANE (0.52) ELANECTSKMEN1KMT2ACYP3A4
SCHEMBL19656274 0.87 ELANE (0.49) ELANECTSKMEN1KMT2ACYP3A4
SCHEMBL19656260 0.86 ELANE (0.49) ELANECTSKMEN1KMT2ACYP3A4
SCHEMBL19640000 0.85 ELANE (0.56) ELANECTSKMEN1KMT2ACYP3A4
SCHEMBL19656244 0.84 ELANE (0.47) ELANECTSKMEN1KMT2ACYP2C9
SCHEMBL19656262 0.84 ELANE (0.49) ELANECTSKMEN1KMT2A
SCHEMBL21796105 0.84 ELANE (0.49) ELANECTSKMEN1KMT2A
Benzene SCHEMBL19639971 0.83 ELANE (0.48) ELANECTSKMEN1KMT2A
SCHEMBL19656257 0.83 ELANE (0.47) ELANECTSKMEN1KMT2A
SCHEMBL19656245 0.83 ELANE (0.48) ELANEMEN1KMT2ACYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017207432-A1 NOVEL COMPOUNDS CHIESI FARMACEUTICI S.P.A. (IT) 2017-12-07 WO disclosed