SCHEMBL19685979

SCHEMBL19685979

CC1(Nc2ncc3nc(Nc4cc(F)cc(Cl)c4)[nH]c3n2)CCOCC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCDIN3D Q7Z5W3 1/20 0.34
EPAS1 Q99814 2/20 0.34
BUB1 O43683 1/20 0.33
RAPGEF4 Q8WZA2 1/20 0.32
TYRO3 Q06418 4/20 0.32
AXL P30530 2/20 0.32
MERTK Q12866 2/20 0.32
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
MAPK1 P28482 1/20 0.31
OPRL1 P41146 1/20 0.31
GRM4 Q14833 1/20 0.31
SELP P16109 1/20 0.31
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29717657 0.86 GRM4 (0.31) GRM4
SCHEMBL19685543 0.85 GRM5 (0.39) HDAC3HDAC1HDAC2HDAC6CYP3A4
SCHEMBL19685710 0.77 DYRK1A (0.36) HDAC3HDAC1HDAC2HDAC6CYP3A4
SCHEMBL29717707 0.77 LATS1 (0.39)
SCHEMBL19689004 0.76 GRM5 (0.42) HDAC3HDAC1HDAC2HDAC6CYP3A4
SCHEMBL19685999 0.76 GRM5 (0.42) HDAC3HDAC1HDAC2HDAC6CYP3A4
SCHEMBL19665698 0.75 MAPK8 (0.46) MAPK1
SCHEMBL29802855 0.75 MAPK8 (0.46) MAPK1
SCHEMBL21385847 0.74 MAPK8 (0.46) MAPK1
SCHEMBL19666607 0.72 MAPK8 (0.44) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017210408-A1 ANIMAL AND HUMAN ANTI-TRYPANOSOMONAL AND ANTI-LEISHMANIA AGENTS CELGENE CORPORATION (US) 2017-12-07 WO disclosed