SCHEMBL1970533

SCHEMBL1970533

CN(C(=O)N(C)[C@@H]1CN(C(=O)[C@H]2CC[C@H](C(=O)O)CC2)C[C@H]1c1ccc(F)cc1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.81

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 20/20 0.81
TACR2 P21452 12/20 0.81
TACR3 P29371 11/20 0.78
TAC3 Q9UHF0 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1970534 1.00 TACR1 (0.81) TACR1TACR2TACR3TAC3
SCHEMBL1971934 0.93 TACR1 (0.79) TACR1TACR2TACR3TAC3
SCHEMBL1973394 0.93 TACR1 (0.79) TACR1TACR2TACR3TAC3
SCHEMBL1971935 0.93 TACR1 (0.79) TACR1TACR2TACR3TAC3
SCHEMBL1966913 0.93 TACR1 (0.81) TACR1TACR2TACR3TAC3
SCHEMBL1966911 0.93 TACR1 (0.81) TACR1TACR2TACR3TAC3
SCHEMBL1969658 0.93 TACR1 (0.90) TACR1TACR2TACR3TAC3
SCHEMBL1968121 0.92 TACR1 (0.80) TACR1TACR2TACR3
SCHEMBL1968119 0.92 TACR1 (0.80) TACR1TACR2TACR3
SCHEMBL1968740 0.92 TACR1 (0.80) TACR1TACR2TACR3TAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2336105-B9 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME TAKEDA PHARMACEUTICAL (JP) 2014-09-17 EP disclosed
EP-2336105-B1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME TAKEDA PHARMACEUTICAL (JP) 2014-02-12 EP disclosed
EP-2336105-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME Takeda Pharmaceutical Company Limited (JP) 2011-06-22 EP disclosed