SCHEMBL19720490

SCHEMBL19720490

Cn1nc(Br)cc1N1CCC(O)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PHGDH O43175 1/20 0.36
IRAK1 P51617 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.35
CNR2 P34972 9/20 0.34
PDE10A Q9Y233 1/20 0.34
AR P10275 1/20 0.34
SUV39H2 Q9H5I1 1/20 0.34
C5AR1 P21730 1/20 0.33
SMPD3 Q9NY59 2/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
GLA P06280 1/20 0.32
POLB P06746 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
RECQL P46063 1/20 0.32
KMT2A Q03164 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16141508 1.00 PHGDH (0.36) PHGDHIRAK1IRAK4CNR2PDE10A
SCHEMBL17473423 1.00 PHGDH (0.36) PHGDHIRAK1IRAK4CNR2PDE10A
SCHEMBL17473353 0.79 PDE10A (0.36) PDE10A
SCHEMBL17473468 0.79 MAPK8 (0.43)
SCHEMBL16141527 0.79 MAPK8 (0.43)
SCHEMBL16141509 0.79 PDE10A (0.36) PDE10A
SCHEMBL17473357 0.79 MAPK8 (0.43)
SCHEMBL16141450 0.76 PDE10A (0.34) PDE10A
SCHEMBL16141548 0.74 EGLN2 (0.41) KDM4EALDH1A1
SCHEMBL17473421 0.74 HRH3 (0.46) LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2980089-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2017-12-20 EP disclosed