SCHEMBL1973100

SCHEMBL1973100

CN(Cc1ccc(Cl)cc1)C(=O)OC1(N)CCN(c2ncnc3[nH]ccc23)CC1

nearest known ligand 0.76

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 20/20 0.76
AKT2 P31751 13/20 0.76
ROCK2 O75116 12/20 0.62
AKT3 Q9Y243 10/20 0.62
KCNH2 Q12809 7/20 0.62
CYP2C9 P11712 2/20 0.62
CYP2D6 P10635 1/20 0.60
RPS6KB1 P23443 1/20 0.60
GSK3B P49841 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1002157 0.86 AKT1 (1.00) AKT1AKT2ROCK2AKT3KCNH2
SCHEMBL16105745 0.83 AKT2 (0.76) AKT1AKT2ROCK2AKT3KCNH2
SCHEMBL1001932 0.77 AKT2 (0.75) AKT1AKT2ROCK2AKT3KCNH2
SCHEMBL1001031 0.77 AKT2 (1.00) AKT1AKT2ROCK2AKT3KCNH2
SCHEMBL1002126 0.76 AKT2 (1.00) AKT1AKT2ROCK2AKT3KCNH2
SCHEMBL29367023 0.76 AKT2 (1.00) AKT1AKT2ROCK2AKT3KCNH2
SCHEMBL3655624 0.76 AKT1 (0.64) AKT1AKT2ROCK2AKT3KCNH2
SCHEMBL15809745 0.75 AKT1 (0.77) AKT1AKT2ROCK2AKT3KCNH2
SCHEMBL392420 0.75 AKT1 (1.00) AKT1AKT2ROCK2AKT3KCNH2
SCHEMBL1973751 0.75 AKT2 (0.77) AKT1AKT2ROCK2AKT3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1812004-B1 ORTHO- CONDENSED PYRIDINE AND PYRIMIDINE DERIVATIVES (E. G. PURINES) AS PROTEIN KINASES INHIBITORS ASTEX THERAPEUTICS LTD (GB) 2011-06-22 EP claimed