SCHEMBL19733249

SCHEMBL19733249

C[C@]12CCC[C@H]1[C@@H]1CC[C@@H]3C[C@H](OS(=O)(=O)O[C@@H]4CC[C@H]5[C@H](CC[C@@H]6[C@H]5CC[C@@]5(C)CCC[C@@H]65)C4)CC[C@@H]3[C@@H]1CC2

nearest known ligand 0.81

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 14/20 0.81
GRIN2B Q13224 14/20 0.81
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
NR1I3 Q14994 1/20 0.36
STS P08842 1/20 0.33
GRIN2D O15399 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2C Q14957 1/20 0.32
MBOAT4 Q96T53 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19253188 1.00 GRIN1 (0.81) GRIN1GRIN2BCDK5CDK5R1NR1I3
SCHEMBL19253189 0.90 GRIN1 (1.00) GRIN1GRIN2BGRIN2DGRIN2AGRIN2C
SCHEMBL6853527 0.83 GRIN1 (0.68) GRIN1GRIN2BCDK5CDK5R1NR1I3
SCHEMBL4605996 0.81 GRIN1 (0.68) GRIN1GRIN2BCDK5CDK5R1NR1I3
SCHEMBL1325195 0.80 GRIN1 (0.67) GRIN1GRIN2BCDK5CDK5R1NR1I3
SCHEMBL19253181 0.77 GRIN1 (0.82) GRIN1GRIN2BCDK5CDK5R1NR1I3
SCHEMBL19253232 0.77 GRIN1 (0.82) GRIN1GRIN2BCDK5CDK5R1NR1I3
SCHEMBL19733259 0.77 GRIN1 (0.82) GRIN1GRIN2BCDK5CDK5R1NR1I3
SCHEMBL19253162 0.77 GRIN1 (0.82) GRIN1GRIN2BCDK5CDK5R1NR1I3
SCHEMBL30645499 0.76 GRIN1 (0.58) GRIN1GRIN2BCDK5CDK5R1NR1I3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3260462-A1 AMPHIPHILIC COMPOUNDS WITH NEUROPROTECTIVE PROPERTIES Ustav Organicke Chemie A Biochemie Av Cr, V.v.i. (CZ) 2017-12-27 EP disclosed