SCHEMBL1973541

SCHEMBL1973541

NC1(OC(=O)NCc2ccc(C(F)(F)F)cc2)CCN(c2ncnc3[nH]ccc23)CC1

nearest known ligand 0.77

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKT2 P31751 16/20 0.77
AKT1 P31749 4/20 0.60
CYP2C9 P11712 3/20 0.60
ROCK2 O75116 2/20 0.60
KCNH2 Q12809 1/20 0.60
AKT3 Q9Y243 1/20 0.60
KIT P10721 1/20 0.54
JAK2 O60674 2/20 0.50
JAK1 P23458 2/20 0.50
TYK2 P29597 2/20 0.50
JAK3 P52333 2/20 0.50
CYP2D6 P10635 1/20 0.48
RPS6KB1 P23443 1/20 0.48
GSK3B P49841 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1975450 0.90 AKT2 (0.80) AKT2AKT1CYP2C9ROCK2KCNH2
SCHEMBL16105745 0.88 AKT2 (0.76) AKT2AKT1CYP2C9ROCK2KCNH2
SCHEMBL1001963 0.87 AKT2 (1.00) AKT2AKT1CYP2C9ROCK2KCNH2
SCHEMBL1974534 0.82 AKT2 (0.77) AKT2AKT1CYP2C9ROCK2KCNH2
SCHEMBL1968905 0.81 AKT2 (0.61) AKT2AKT1CYP2C9ROCK2KCNH2
SCHEMBL1975865 0.80 AKT2 (0.76) AKT2AKT1CYP2C9ROCK2KCNH2
SCHEMBL1970926 0.79 AKT2 (0.77) AKT2AKT1CYP2C9ROCK2KCNH2
SCHEMBL1973751 0.78 AKT2 (0.77) AKT2AKT1CYP2C9ROCK2KCNH2
SCHEMBL1003173 0.78 AKT2 (1.00) AKT2AKT1CYP2C9ROCK2KCNH2
SCHEMBL1002396 0.78 AKT2 (1.00) AKT2AKT1CYP2C9ROCK2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1812004-B1 ORTHO- CONDENSED PYRIDINE AND PYRIMIDINE DERIVATIVES (E. G. PURINES) AS PROTEIN KINASES INHIBITORS ASTEX THERAPEUTICS LTD (GB) 2011-06-22 EP claimed