SCHEMBL19746465

SCHEMBL19746465

O=c1cc(-c2noc(C(F)(F)F)n2)ccn1Cc1ccc2ncccc2c1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 18/20 0.51
HDAC1 Q13547 13/20 0.47
HDAC8 Q9BY41 7/20 0.47
MET P08581 1/20 0.45
HDAC4 P56524 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19746290 0.89 HDAC6 (0.48) HDAC6HDAC1HDAC8HDAC4
SCHEMBL19747081 0.87 HDAC6 (0.61) HDAC6HDAC1HDAC8HDAC4
SCHEMBL19747484 0.87 HDAC6 (0.56) HDAC6HDAC1HDAC8HDAC4
SCHEMBL19746485 0.86 HDAC6 (0.52) HDAC6HDAC1HDAC8
SCHEMBL19746017 0.84 HDAC6 (0.50) HDAC6HDAC1HDAC8HDAC4
SCHEMBL19746460 0.83 HDAC6 (0.46) HDAC6HDAC1HDAC8HDAC4
SCHEMBL19746136 0.82 HDAC6 (0.57) HDAC6HDAC1HDAC8HDAC4
SCHEMBL19746127 0.82 HDAC6 (0.46) HDAC6HDAC1HDAC8HDAC4
SCHEMBL19746376 0.81 HDAC6 (0.50) HDAC6HDAC1HDAC8HDAC4
SCHEMBL19746691 0.81 HDAC6 (0.56) HDAC6HDAC1HDAC8HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017222952-A1 3- HETEROARYL SUBSTITUTED 5-TRIFLUOROMETHYL OXADIAZOLES AS HISTONE DEACETYLASE 6 (HDAC6) INHIBITORS MERCK SHARP & DOHME CORP. (US) 2017-12-28 WO claimed