SCHEMBL19746575

SCHEMBL19746575

Cc1cnc(Cn2ccc(-c3noc(C(F)(F)F)n3)cc2=O)cn1

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 20/20 0.60
HDAC1 Q13547 18/20 0.60
HDAC8 Q9BY41 7/20 0.49
HDAC5 Q9UQL6 4/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19746593 0.86 HDAC6 (0.45) HDAC6HDAC1HDAC8
SCHEMBL19746639 0.85 HDAC6 (0.47) HDAC6HDAC1HDAC8HDAC5
SCHEMBL19747353 0.84 HDAC6 (0.58) HDAC6HDAC1HDAC8
SCHEMBL19746962 0.84 HDAC6 (0.55) HDAC6HDAC1HDAC8HDAC5
SCHEMBL19746864 0.83 HDAC6 (0.46) HDAC6HDAC1HDAC8HDAC5
SCHEMBL19747014 0.80 HDAC6 (0.44) HDAC6HDAC1HDAC8HDAC5
SCHEMBL19746485 0.80 HDAC6 (0.52) HDAC6HDAC1HDAC8HDAC5
SCHEMBL19746081 0.80 HDAC6 (0.47) HDAC6HDAC1HDAC8HDAC5
SCHEMBL19747433 0.80 HDAC6 (0.42) HDAC6HDAC1HDAC8
SCHEMBL19746707 0.80 HDAC6 (0.60) HDAC6HDAC1HDAC8HDAC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017222952-A1 3- HETEROARYL SUBSTITUTED 5-TRIFLUOROMETHYL OXADIAZOLES AS HISTONE DEACETYLASE 6 (HDAC6) INHIBITORS MERCK SHARP & DOHME CORP. (US) 2017-12-28 WO claimed