SCHEMBL19772098

SCHEMBL19772098

C[C@@H](c1ccc(C(F)(F)F)cc1F)C(C)(C)C

nearest known ligand 0.69

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 18/20 0.69
IDO1 P14902 1/20 0.38
CYP3A4 P08684 1/20 0.37
CYP3A5 P20815 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19771904 1.00 PDE2A (0.69) PDE2AIDO1CYP3A4CYP3A5
SCHEMBL22389476 0.85 PDE2A (0.54) PDE2AIDO1
SCHEMBL22389494 0.85 PDE2A (0.54) PDE2AIDO1
SCHEMBL84521 0.82 PDE2A (0.70) PDE2AIDO1CYP3A4CYP3A5
SCHEMBL1035450 0.81 PDE2A (1.00) PDE2A
SCHEMBL20811535 0.80 PDE2A (0.67) PDE2AIDO1
SCHEMBL22221342 0.80 PDE2A (0.67) PDE2AIDO1
SCHEMBL20811529 0.80 PDE2A (0.67) PDE2AIDO1
SCHEMBL18103269 0.79 PDE2A (0.66) PDE2AIDO1CYP3A4CYP3A5
SCHEMBL3315570 0.79 PDE2A (0.66) PDE2AIDO1CYP3A4CYP3A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9868748-B2 Thiazolopyrrolidine inhibitors of ROR- γ VITAE PHARMACEUTICALS, INC. (US) 2018-01-16 US disclosed