SCHEMBL19781776

SCHEMBL19781776

CC(C)Oc1ccc(-c2cnc3ccc(-c4ccc(O)cc4)cn23)cc1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FYN P06241 12/20 0.54
MKNK1 Q9BUB5 3/20 0.46
MKNK2 Q9HBH9 3/20 0.46
CLK1 P49759 1/20 0.46
RIPK2 O43353 1/20 0.43
PIK3CA P42336 1/20 0.42
MTOR P42345 1/20 0.42
KCNH2 Q12809 1/20 0.41
CYP1A2 P05177 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19781539 0.93 CLK1 (0.47) FYNMKNK1MKNK2CLK1RIPK2
SCHEMBL24460223 0.87 BCL2 (0.44) FYNMKNK1MKNK2CLK1PIK3CA
SCHEMBL19781775 0.87 FLT3 (0.51) FYNMKNK1CLK1PIK3CAMTOR
SCHEMBL19781168 0.87 SCN5A (0.50) FYNMKNK1MKNK2CLK1RIPK2
SCHEMBL19781553 0.87 SCN5A (0.50) FYNMKNK1MKNK2CLK1RIPK2
SCHEMBL19781132 0.85 CLK1 (0.48) FYNMKNK1MKNK2CLK1KCNH2
SCHEMBL19781151 0.85 CLK1 (0.48) FYNMKNK1MKNK2CLK1KCNH2
SCHEMBL19781183 0.85 KMT2A (0.54) FYNMKNK1MKNK2CLK1
SCHEMBL19781173 0.85 CLK1 (0.43) FYNMKNK1MKNK2CLK1RIPK2
SCHEMBL19781610 0.85 CLK1 (0.43) FYNMKNK1MKNK2CLK1RIPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230303569-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS ARISAN THERAPEUTICS INC. (US) 2023-09-28 US disclosed
US-20230303569-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS ARISAN THERAPEUTICS INC. (US) 2023-09-28 US disclosed
US-20230303569-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS ARISAN THERAPEUTICS INC. (US) 2023-09-28 US disclosed
US-20220193038-A1 COMPOUNDS FOR THE TREATMENT OF ARENAVIRUS INFECTION ARISAN THERAPEUTICS INC. (US) 2022-06-23 US disclosed
US-11352328-B2 Heterocyclic compounds for the treatment of arenavirus ARISAN THERAPEUTICS INC. (US) 2022-06-07 US disclosed
WO-2022108849-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS ARISAN THERAPEUTICS INC. (US) 2022-05-27 WO disclosed
WO-2020117794-A1 COMPOUNDS FOR THE TREATMENT OF ARENAVIRUS INFECTION ARISAN THERAPEUTICS, INC. (US) 2020-06-11 WO disclosed
US-20190308938-A1 Heterocyclic Compounds for the Treatment of Arenavirus NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2019-10-10 US disclosed
WO-2018013430-A2 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF ARENAVIRUS INFECTION ARISAN THERAPEUTICS INC. (US) 2018-01-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220193038-A1 COMPOUNDS FOR THE TREATMENT OF ARENAVIRUS INFECTION HAVCR2, ZC3HAV1, CD4 FYN 1552/4885MKNK1 2116/4885MKNK2 2340/4885
US-20230303569-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS C3AR1, C9, C1R FYN 1748/4885MKNK1 3245/4885MKNK2 3215/4885
US-11352328-B2 Heterocyclic compounds for the treatment of arenavirus C9, C1R, C1S FYN 1982/4885MKNK1 3509/4885MKNK2 3686/4885
US-20190308938-A1 Heterocyclic Compounds for the Treatment of Arenavirus C9, C1R, C1S FYN 1982/4885MKNK1 3509/4885MKNK2 3686/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.