SCHEMBL19783378

SCHEMBL19783378

COc1cc(Br)c2nc(NC(=O)OC(C)(C)C)sc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 10/20 0.52
HSD17B10 Q99714 2/20 0.44
RAB9A P51151 4/20 0.43
NPC1 O15118 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
DYRK1A Q13627 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTT P42858 1/20 0.43
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
SENP6 Q9GZR1 1/20 0.43
TSHR P16473 1/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TP53 P04637 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30189684 1.00 LCK (0.52) LCKHSD17B10RAB9ANPC1SMN1; SMN2
SCHEMBL19630817 0.88 LCK (0.54) LCKRAB9ANPC1DYRK1ACYP1A2
SCHEMBL2274858 0.86 LCK (0.61) LCKKDM4EALDH1A1MAPT
SCHEMBL19630789 0.85 LCK (0.52) LCKRAB9ANPC1SMN1; SMN2HTT
SCHEMBL2918251 0.83 LCK (0.50) LCKRAB9A
SCHEMBL2920108 0.83 LCK (0.50) LCKRAB9AMAPT
SCHEMBL2918417 0.83 LCK (0.54) LCKRAB9A
SCHEMBL30189854 0.83 LCK (0.48) LCKRAB9ANPC1SMN1; SMN2DYRK1A
SCHEMBL19783377 0.83 LCK (0.48) LCKRAB9ANPC1SMN1; SMN2DYRK1A
SCHEMBL2920743 0.82 LCK (0.49) LCKRAB9ADYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
WO-2018013774-A1 BICYCLIC HETEROARYL SUBSTITUTED COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-01-18 WO disclosed