SCHEMBL19785230

SCHEMBL19785230

Cc1nccc(Sc2ncc(N3CCC4(CCC[C@H]4N)CC3)nc2C2CC2)c1Cl

nearest known ligand 0.67

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 20/20 0.67
KCNH2 Q12809 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19785479 0.91 PTPN11 (0.80) PTPN11KCNH2
SCHEMBL19785110 0.85 PTPN11 (0.80) PTPN11
SCHEMBL19785227 0.84 PTPN11 (0.81) PTPN11KCNH2
SCHEMBL19785229 0.84 PTPN11 (0.84) PTPN11KCNH2
SCHEMBL30511929 0.84 PTPN11 (0.84) PTPN11KCNH2
SCHEMBL25514142 0.83 PTPN11 (0.65) PTPN11
SCHEMBL16914407 0.81 PTPN11 (1.00) PTPN11KCNH2
SCHEMBL16914264 0.80 PTPN11 (1.00) PTPN11
SCHEMBL19785225 0.79 PTPN11 (0.78) PTPN11KCNH2
SCHEMBL23186805 0.79 PTPN11 (0.69) PTPN11KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018013597-A1 2,5-DISUBSTITUTED 3-METHYL PYRAZINES AND 2,5,6-TRISUBSTITUTED 3-METHYL PYRAZINES AS ALLOSTERIC SHP2 INHIBITORS Revolution Medicines, Inc. (US) 2018-01-18 WO disclosed