SCHEMBL19785267

SCHEMBL19785267

Cc1nc(N2CCC3(CCCC3)CC2)c(CO)nc1Sc1cccc2cc[nH]c12

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 15/20 0.42
KCNH2 Q12809 2/20 0.35
EGFR P00533 1/20 0.35
SCN10A Q9Y5Y9 1/20 0.33
HTR1A P08908 1/20 0.31
HTR1D P28221 1/20 0.31
HTR1B P28222 1/20 0.31
KIF18A Q8NI77 1/20 0.31
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23186865 0.83 PTPN11 (0.52) PTPN11KCNH2EGFR
SCHEMBL23186812 0.81 PTPN11 (0.49) PTPN11KCNH2EGFR
SCHEMBL23186809 0.81 PTPN11 (0.46) PTPN11KCNH2EGFR
SCHEMBL23186864 0.81 PTPN11 (0.39) PTPN11KCNH2EGFRSCN10A
SCHEMBL23186828 0.79 PTPN11 (0.41) PTPN11KCNH2EGFR
SCHEMBL21154444 0.76 PTPN11 (0.58) PTPN11KCNH2EGFR
SCHEMBL23186853 0.75 PTPN11 (0.71) PTPN11
SCHEMBL23186859 0.74 PTPN11 (0.39) PTPN11KIF18A
SCHEMBL19785059 0.74 PTPN11 (0.50) PTPN11KCNH2
SCHEMBL19785588 0.73 PTPN11 (0.55) PTPN11KCNH2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018013597-A1 2,5-DISUBSTITUTED 3-METHYL PYRAZINES AND 2,5,6-TRISUBSTITUTED 3-METHYL PYRAZINES AS ALLOSTERIC SHP2 INHIBITORS Revolution Medicines, Inc. (US) 2018-01-18 WO disclosed