SCHEMBL19785644

SCHEMBL19785644

COc1ccc(SC/C=C\SSCc2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.44
MAOB P27338 2/20 0.42
MAOA P21397 1/20 0.42
LTA4H P09960 2/20 0.41
ALDH1A1 P00352 3/20 0.39
LMNA P02545 2/20 0.39
MAPT P10636 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
HTT P42858 1/20 0.39
KDM4E B2RXH2 1/20 0.39
TSHR P16473 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
G6PC1 P35575 1/20 0.38
CTSB P07858 1/20 0.38
HDAC3 O15379 1/20 0.37
NCOR1 O75376 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19786132 1.00 APP (0.44) APPMAOBMAOALTA4HALDH1A1
SCHEMBL21190092 0.95 APP (0.44) APPMAOBMAOALTA4HALDH1A1
SCHEMBL21189961 0.95 APP (0.44) APPMAOBMAOALTA4HALDH1A1
SCHEMBL19786028 0.88 APP (0.47) APPMAOBMAOAALDH1A1MAPT
SCHEMBL19785649 0.88 APP (0.47) APPMAOBMAOAALDH1A1MAPT
SCHEMBL21190042 0.87 APP (0.46) APPMAOBMAOAALDH1A1MAPT
SCHEMBL21189918 0.87 APP (0.46) APPMAOBMAOAALDH1A1LMNA
SCHEMBL21189903 0.87 APP (0.46) APPMAOBMAOAALDH1A1LMNA
SCHEMBL21190022 0.87 APP (0.46) APPMAOBMAOAALDH1A1MAPT
SCHEMBL21189901 0.86 MAOB (0.43) MAOBMAOAALDH1A1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019143143-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING NEUROBLASTOMA OR RHEUMATOID ARTHRITIS 숙명여자대학교 산학협력단 2019-07-25 WO disclosed
WO-2019143142-A1 NOVEL PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING GLIOBLASTOMA 숙명여자대학교 산학협력단 2019-07-25 WO disclosed
WO-2018012947-A1 NOVEL ORGANIC SULFUR COMPOUND, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING CANCER OR AN INFLAMMATORY DISEASE, CONTAINING SAME AS ACTIVE INGREDIENT 숙명여자대학교 산학협력단 2018-01-18 WO disclosed