SCHEMBL19787604

SCHEMBL19787604

COc1cc(N2C[C@H]3C[C@@H](C2)[C@@H]3N)ccn1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 3/20 0.43
CHRM2 P08172 1/20 0.42
SMARCA2 P51531 2/20 0.41
SMARCA4 P51532 2/20 0.41
PSEN1 P49768 4/20 0.41
PSEN2 P49810 4/20 0.41
APH1B Q8WW43 4/20 0.41
NCSTN Q92542 4/20 0.41
APH1A Q96BI3 4/20 0.41
PSENEN Q9NZ42 4/20 0.41
LOX P28300 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.41
NR1H2 P55055 1/20 0.40
NR1H3 Q13133 1/20 0.40
CYP17A1 P05093 3/20 0.40
APP P05067 2/20 0.39
CHRM1 P11229 1/20 0.35
NTRK1 P04629 1/20 0.35
ACACB O00763 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21069145 0.93 PSEN1 (0.45) CHRM4CHRM2SMARCA2SMARCA4PSEN1
SCHEMBL21374488 0.93 PSEN1 (0.45) CHRM4CHRM2SMARCA2SMARCA4PSEN1
SCHEMBL21050448 0.93 PSEN1 (0.45) CHRM4CHRM2SMARCA2SMARCA4PSEN1
SCHEMBL21050446 0.93 PSEN1 (0.45) CHRM4CHRM2SMARCA2SMARCA4PSEN1
SCHEMBL21050443 0.93 PSEN1 (0.45) CHRM4CHRM2SMARCA2SMARCA4PSEN1
SCHEMBL24083325 0.93 PSEN1 (0.45) CHRM4CHRM2SMARCA2SMARCA4PSEN1
SCHEMBL16685020 0.86 CHRM4 (0.47) CHRM4CHRM2SMARCA2SMARCA4PSEN1
Hydrochloric Acid SCHEMBL17077952 0.85 CHRM4 (0.47) CHRM4CHRM2SMARCA2SMARCA4PSEN1
SCHEMBL31614725 0.80 CHRM4 (0.47) CHRM4CHRM2SMARCA2SMARCA4PSEN1
SCHEMBL20159687 0.80 NR1H2 (0.41) CHRM4CHRM2SMARCA2SMARCA4PSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3484884-B1 FUSED PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2021-01-27 EP disclosed
WO-2018011164-A1 FUSED PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2018-01-18 WO disclosed