SCHEMBL19789212

SCHEMBL19789212

C=C(CCOc1ccc(Nc2nc(C)nc3ccccc23)cc1)OCC

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.52
MAPT P10636 7/20 0.50
KMT2A Q03164 5/20 0.50
NPSR1 Q6W5P4 4/20 0.50
MEN1 O00255 3/20 0.50
GAA P10253 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
NPY1R P25929 1/20 0.50
NPY2R P49146 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
GPR55 Q9Y2T6 1/20 0.50
KDM4E B2RXH2 5/20 0.48
ALDH1A1 P00352 4/20 0.48
POLB P06746 2/20 0.48
HPGD P15428 2/20 0.48
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 2/20 0.48
CYP2C9 P11712 2/20 0.48
CYP2C19 P33261 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19789175 0.95 TP53 (0.51) TP53MAPTKMT2ANPSR1MEN1
SCHEMBL18088085 0.87 TP53 (0.57) TP53MAPTKMT2ANPSR1MEN1
SCHEMBL18088012 0.84 TP53 (0.56) TP53MAPTKMT2ANPSR1MEN1
SCHEMBL24653613 0.84 MAPT (0.54) TP53MAPTKMT2ANPSR1MEN1
SCHEMBL3114887 0.84 KMT2A (0.67) TP53MAPTKMT2ANPSR1MEN1
SCHEMBL18087996 0.83 TP53 (0.55) TP53MAPTKMT2ANPSR1MEN1
SCHEMBL18088102 0.82 TP53 (0.54) TP53MAPTKMT2ANPSR1MEN1
SCHEMBL18088016 0.82 HDAC1 (0.58) TP53MAPTKMT2ANPSR1MEN1
SCHEMBL19789110 0.82 TP53 (0.50) TP53MAPTKMT2ANPSR1MEN1
SCHEMBL19789132 0.81 HDAC1 (0.47) TP53MAPTKMT2ANPSR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3272742-A1 HISTONE DEACETYLASE INHIBITOR, AND PREPARATION METHOD AND USE THEREOF GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2018-01-24 EP disclosed