SCHEMBL1979127

SCHEMBL1979127

CC1(C)CNC(=O)c2cc3ccc(C(=O)Nc4c[nH]c(CC(=O)NC5CCCC5)n4)cc3n21

nearest known ligand 0.68

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RPS6KA2 Q15349 13/20 0.68
MAPKAPK2 P49137 6/20 0.63
RPS6KA3 P51812 1/20 0.55
CLK1 P49759 1/20 0.45
GSK3B P49841 1/20 0.45
MAP3K14 Q99558 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1979620 0.81 RPS6KA2 (1.00) RPS6KA2MAPKAPK2RPS6KA3
SCHEMBL1979125 0.78 RPS6KA2 (0.68) RPS6KA2MAPKAPK2RPS6KA3CLK1GSK3B
SCHEMBL12598642 0.75 RPS6KA2 (1.00) RPS6KA2RPS6KA3
SCHEMBL1979131 0.72 RPS6KA2 (0.81) RPS6KA2MAPKAPK2RPS6KA3
SCHEMBL12598632 0.72 RPS6KA2 (0.73) RPS6KA2MAPKAPK2RPS6KA3
SCHEMBL12598636 0.72 RPS6KA2 (0.71) RPS6KA2RPS6KA3
SCHEMBL3078970 0.71 RPS6KA2 (0.66) RPS6KA2MAPKAPK2RPS6KA3
SCHEMBL3079464 0.71 RPS6KA3 (1.00) RPS6KA2MAPKAPK2RPS6KA3
SCHEMBL1978707 0.70 RPS6KA2 (0.74) RPS6KA2MAPKAPK2RPS6KA3
SCHEMBL1978106 0.70 RPS6KA2 (0.64) RPS6KA2MAPKAPK2RPS6KA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2509980-A1 HETEROCYCLIC COMPOUNDS CONTAINING AN INDOLE CORE Boehringer Ingelheim International GmbH (DE) 2012-10-17 EP disclosed
WO-2011071716-A1 HETEROCYCLIC COMPOUNDS CONTAINING AN INDOLE CORE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-06-16 WO disclosed