SCHEMBL1979271

SCHEMBL1979271

C[C@]1(c2cc(NC(=O)c3ccc(OCC(F)(F)F)cn3)ccc2F)OC(N)=NCC1(F)F

nearest known ligand 0.70

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.70
BACE2 Q9Y5Z0 11/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1982790 0.94 BACE1 (0.68) BACE1BACE2
SCHEMBL1979940 0.89 BACE1 (0.67) BACE1BACE2
SCHEMBL1979498 0.87 BACE1 (0.69) BACE1BACE2
SCHEMBL1980711 0.84 BACE1 (0.63) BACE1BACE2
SCHEMBL1981723 0.83 BACE1 (0.58) BACE1BACE2
SCHEMBL1975338 0.82 BACE1 (1.00) BACE1BACE2
SCHEMBL1978113 0.82 BACE1 (0.68) BACE1BACE2
SCHEMBL1976269 0.81 BACE1 (0.76) BACE1BACE2
Hydrochloric Acid SCHEMBL1979733 0.81 BACE1 (0.67) BACE1BACE2
SCHEMBL15142499 0.81 BACE1 (0.67) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011069934-A1 2-AMINO-5, 5-DIFLUORO-5, 6-DIHYDRO-4H-OXAZINES AS BACE 1 AND/OR BACE 2 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-16 WO claimed
WO-2011069934-A1 2-AMINO-5, 5-DIFLUORO-5, 6-DIHYDRO-4H-OXAZINES AS BACE 1 AND/OR BACE 2 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-16 WO disclosed