SCHEMBL1979326

SCHEMBL1979326

COc1ccc2[nH]c3cnc(-c4cnn(C)c4)cc3c2c1-c1ccc(C(=O)NCC2CCCN2)cc1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SUV39H2 Q9H5I1 2/20 0.45
IKBKB O14920 13/20 0.42
CHEK2 O96017 1/20 0.42
MET P08581 1/20 0.42
CHUK O15111 1/20 0.40
IGF1R P08069 2/20 0.38
ROCK2 O75116 1/20 0.38
ROCK1 Q13464 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12597811 0.93 IKBKB (0.41) SUV39H2IKBKBCHEK2METCHUK
SCHEMBL3725168 0.92 SUV39H2 (0.46) SUV39H2IKBKBCHEK2METCHUK
SCHEMBL1980453 0.88 SUV39H2 (0.43) SUV39H2IKBKBCHEK2METCHUK
SCHEMBL12597421 0.85 IKBKB (0.44) SUV39H2IKBKBCHEK2METCHUK
SCHEMBL473674 0.85 IKBKB (0.40) SUV39H2IKBKBCHEK2METCHUK
SCHEMBL473788 0.85 IKBKB (0.43) SUV39H2IKBKBCHEK2METCHUK
SCHEMBL3723523 0.85 IKBKB (0.43) SUV39H2IKBKBCHEK2METCHUK
SCHEMBL11908837 0.85 SUV39H2 (0.44) SUV39H2IKBKBCHEK2METCHUK
SCHEMBL12597220 0.83 TLR7 (0.41) IGF1R
SCHEMBL3723610 0.83 HDAC4 (0.42) SUV39H2IKBKBCHEK2METCHUK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed