SCHEMBL1979378

SCHEMBL1979378

NC1c2cccc(F)c2OCC1O

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.37
TAAR1 Q96RJ0 2/20 0.37
CYP2D6 P10635 1/20 0.37
KDM1A O60341 2/20 0.37
KDM1B Q8NB78 1/20 0.37
CA2 P00918 1/20 0.36
ADRA2A P08913 1/20 0.36
TERT O14746 1/20 0.35
HTR2C P28335 2/20 0.34
HTR2B P41595 2/20 0.34
ACHE P22303 1/20 0.31
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1979379 1.00 CYP19A1 (0.37) CYP19A1TAAR1CYP2D6KDM1AKDM1B
SCHEMBL13834855 1.00 CYP19A1 (0.37) CYP19A1TAAR1CYP2D6KDM1AKDM1B
SCHEMBL6900041 1.00 CYP19A1 (0.37) CYP19A1TAAR1CYP2D6KDM1AKDM1B
SCHEMBL6899312 0.80 PSMB8 (0.39) TAAR1CA2ADRA2AHTR2CHTR2B
SCHEMBL2593064 0.79 CYP19A1 (0.41) CYP19A1TAAR1CYP2D6KDM1AKDM1B
SCHEMBL31278211 0.79 KDM1A (0.41) CYP19A1TAAR1CYP2D6KDM1AKDM1B
Hydrochloric Acid SCHEMBL30989938 0.77 KDM1A (0.40) CYP19A1TAAR1CYP2D6KDM1AKDM1B
SCHEMBL6900223 0.77 KDM1A (0.32) KDM1AKDM1B
SCHEMBL13834925 0.77 KDM1A (0.32) KDM1AKDM1B
SCHEMBL13834753 0.74 UGT2B17 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2509950-A1 5-AMINO- 4-HYDROXYPENTOYL AMIDES Janssen R&D Ireland (IE) 2012-10-17 EP disclosed
WO-2011070131-A1 5-AMINO- 4-HYDROXYPENTOYL AMIDES TIBOTEC PHARMACEUTICALS (IE) 2011-06-16 WO disclosed