SCHEMBL1979385

SCHEMBL1979385

COc1ccc(C(NC2=NCC(F)(F)[C@@](C)(c3cc(N=C(c4ccccc4)c4ccccc4)ccc3F)O2)(c2ccccc2)c2ccc(OC)cc2)cc1

nearest known ligand 0.37

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.32
BACE2 Q9Y5Z0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1979501 0.87 BACE1 (0.31) BACE1BACE2
SCHEMBL1980432 0.85 BACE1 (0.33) BACE1
SCHEMBL1977445 0.83 BACE1 (0.40) BACE1BACE2
SCHEMBL1977447 0.83 BACE1 (0.40) BACE1BACE2
SCHEMBL1975419 0.82 BACE1 (0.34) BACE1BACE2
SCHEMBL1975420 0.82 BACE1 (0.34) BACE1BACE2
SCHEMBL14127533 0.82
SCHEMBL13859332 0.81
SCHEMBL2589584 0.79 BACE1 (0.37) BACE1BACE2
SCHEMBL2589589 0.79 BACE1 (0.37) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2509965-A1 2-AMINO-5, 5-DIFLUORO-5, 6-DIHYDRO-4H-OXAZINES AS BACE 1 AND/OR BACE 2 INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-10-17 EP disclosed
WO-2011069934-A1 2-AMINO-5, 5-DIFLUORO-5, 6-DIHYDRO-4H-OXAZINES AS BACE 1 AND/OR BACE 2 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-16 WO disclosed