SCHEMBL1980888

SCHEMBL1980888

CC1(C)N=C(N)O[C@](C)(c2cc(NC(=O)c3ncc(Cl)cc3F)ccc2F)C1(F)F

nearest known ligand 0.66

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.66
BACE2 Q9Y5Z0 10/20 0.65
CYP2D6 P10635 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1981020 0.94 BACE1 (0.67) BACE1BACE2CYP2D6
Hydrochloric Acid SCHEMBL1979781 0.93 BACE1 (0.66) BACE1BACE2CYP2D6
SCHEMBL1981784 0.89 BACE1 (0.69) BACE1BACE2
SCHEMBL1980393 0.89 BACE1 (0.65) BACE1BACE2
SCHEMBL1974548 0.86 BACE1 (0.65) BACE1BACE2CYP2D6
SCHEMBL1974551 0.86 BACE1 (0.65) BACE1BACE2CYP2D6
SCHEMBL1980007 0.86 BACE1 (0.68) BACE1BACE2CYP2D6
SCHEMBL1979083 0.85 BACE1 (0.69) BACE1BACE2
Hydrochloric Acid SCHEMBL1981515 0.85 BACE1 (0.67) BACE1BACE2CYP2D6
Hydrochloric Acid SCHEMBL1980454 0.84 BACE1 (0.68) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011069934-A1 2-AMINO-5, 5-DIFLUORO-5, 6-DIHYDRO-4H-OXAZINES AS BACE 1 AND/OR BACE 2 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-16 WO disclosed