Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL1983246

COc1cc(C(C)(C)c2cnc(SCc3c(F)cc(N[C@H]4CC[N+](C)(Cc5ccc(F)cc5)C4)cc3Cl)n2-c2ccc(F)cc2)ccc1Cl.O=C([O-])C(F)(F)F

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 19/20 0.51
NR1H4 Q96RI1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL1983249 0.91 GPBAR1 (0.49) GPBAR1
Trifluoroacetic Acid SCHEMBL1986610 0.91 GPBAR1 (0.52) GPBAR1NR1H4
SCHEMBL15380423 0.88 GPBAR1 (0.53) GPBAR1
SCHEMBL13270245 0.87 GPBAR1 (0.55) GPBAR1NR1H4
Trifluoroacetic Acid SCHEMBL15380567 0.83 GPBAR1 (0.53) GPBAR1
Trifluoroacetic Acid SCHEMBL15380288 0.83 GPBAR1 (0.51) GPBAR1
Trifluoroacetic Acid SCHEMBL15380565 0.82 GPBAR1 (0.52) GPBAR1
Trifluoroacetic Acid SCHEMBL15380566 0.82 GPBAR1 (0.52) GPBAR1
SCHEMBL12593304 0.80 GPBAR1 (0.56) GPBAR1NR1H4
SCHEMBL15380775 0.80 GPBAR1 (0.56) GPBAR1NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2509960-A1 TGR5 AGONISTS Exelixis, Inc. (US) 2012-10-17 EP disclosed
WO-2011071565-A1 TGR5 AGONISTS EXELIXIS, INC. (US) 2011-06-16 WO disclosed