SCHEMBL19853560

SCHEMBL19853560

NS(=O)(=O)c1ccccc1-c1ccc(C(=O)Nc2ccccc2Oc2cc3ccccc3cc2C(=O)OCc2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
F10 P00742 20/20 0.57
KLK1 P06870 2/20 0.57
PLG P00747 1/20 0.57
PLAT P00750 1/20 0.57
PRSS1 P07477 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12133149 0.88 F10 (0.62) F10KLK1PLGPLATPRSS1
SCHEMBL12133152 0.88 F10 (0.64) F10KLK1PLGPLATPRSS1
SCHEMBL12133160 0.86 F10 (0.67) F10KLK1PLGPLATPRSS1
SCHEMBL12132434 0.81 F10 (0.65) F10KLK1PLGPLATPRSS1
SCHEMBL12133153 0.81 F10 (0.57) F10KLK1PLGPLATPRSS1
SCHEMBL18772846 0.79 F10 (0.74) F10KLK1PLGPLATPRSS1
SCHEMBL890638 0.78 F10 (0.67) F10KLK1PLGPLATPRSS1
SCHEMBL890995 0.78 F10 (0.74) F10KLK1PLGPLATPRSS1
SCHEMBL15063394 0.76 F10 (0.62) F10KLK1PLGPLATPRSS1
SCHEMBL898836 0.74 F10 (0.70) F10KLK1PLGPLATPRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10179124-B2 Benzamides and related inhibitors of factor Xa MILLENNIUM PHARMACEUTICALS, INC. (US) 2019-01-15 US disclosed
US-20180036296-A1 BENZAMIDES AND RELATED INHIBITORS OF FACTOR XA COR THERAPEUTICS, INC. 2018-02-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180036296-A1 BENZAMIDES AND RELATED INHIBITORS OF FACTOR XA TFPI, F12, TFPI2 F10 13/4885KLK1 637/4885PLG 18/4885
US-10179124-B2 Benzamides and related inhibitors of factor Xa TFPI, F12, TFPI2 F10 13/4885KLK1 637/4885PLG 18/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.