SCHEMBL19859005

SCHEMBL19859005

COC(=O)c1ccc(Cl)cc1OCCN1CCCC1

nearest known ligand 0.63

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.63
MEN1 O00255 1/20 0.63
KMT2A Q03164 1/20 0.63
KDM4E B2RXH2 3/20 0.53
HRH3 Q9Y5N1 1/20 0.52
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
LTA4H P09960 2/20 0.49
PTGS2 P35354 1/20 0.49
POLB P06746 1/20 0.48
TSHR P16473 1/20 0.48
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19859001 0.99 GAA (0.65) GAAMEN1KMT2AKDM4EHRH3
SCHEMBL19859010 0.89 TSHR (0.64) GAAMEN1KMT2AKDM4ENPC1
SCHEMBL19859086 0.88 MEN1 (0.50) GAAMEN1KMT2AKDM4EHRH3
SCHEMBL19870511 0.87 MEN1 (0.49) GAAMEN1KMT2AKDM4EHRH3
SCHEMBL19869220 0.86 KDM4E (0.56) MEN1KMT2AKDM4EHRH3NPC1
SCHEMBL19859017 0.85 KDM4E (0.58) MEN1KMT2AKDM4EHRH3NPC1
SCHEMBL954407 0.82 MEN1 (0.90) GAAMEN1KMT2AKDM4ESMN1; SMN2
SCHEMBL6042774 0.81 MEN1 (0.61) GAAMEN1KMT2AKDM4EPOLB
SCHEMBL21750480 0.81 MEN1 (0.93) GAAMEN1KMT2AKDM4ESMN1; SMN2
SCHEMBL19859009 0.80 ABL1 (0.54) KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018029604-A1 C-3 NOVEL TRITERPENONE WITH C-17 REVERSE AMIDE DERIVATIVES AS HIV INHIBITORS HETERO LABS LIMITED (IN) 2018-02-15 WO disclosed
WO-2018029604-A1 C-3 NOVEL TRITERPENONE WITH C-17 REVERSE AMIDE DERIVATIVES AS HIV INHIBITORS HETERO LABS LIMITED (IN) 2018-02-15 WO disclosed