SCHEMBL19861356

SCHEMBL19861356

C/C=C/C[C@@H](C)C[C@H]1C(=O)N[C@@H](CC)C(=O)N(C)[C@H](CSCCN(CC)CC)C(=O)N(C)[C@@H](CC(C)(C)O)C(=O)N[C@H](C(C)C)C(=O)N(C)[C@H](CC(C)C)C(=O)N[C@H](C)C(=O)N[C@@H](C)C(=O)N(C)[C@@H](CC(C)C)C(=O)N(C)[C@@H](CCC(C)C)C(=O)N(C)[C@@H](C(C)C)C(=O)N1C

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPIA P62937 19/20 0.71
PPIB P23284 8/20 0.64
CYP3A4 P08684 2/20 0.64
CYP2C9 P11712 2/20 0.64
PPIF P30405 2/20 0.64
CYP2C19 P33261 2/20 0.64
ABCB1 P08183 3/20 0.60
SLCO1B1 Q9Y6L6 3/20 0.56
ABCB11 O95342 2/20 0.56
ABCC2 Q92887 2/20 0.56
SLCO1B3 Q9NPD5 2/20 0.56
MEN1 O00255 1/20 0.53
NPC1 O15118 1/20 0.53
ABCC3 O15438 1/20 0.53
GMNN O75496 1/20 0.53
USP2 O75604 1/20 0.53
SLCO2B1 O94956 1/20 0.53
LMNA P02545 1/20 0.53
POLB P06746 1/20 0.53
MAPT P10636 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20076272 0.96 PPIA (0.66) PPIAPPIBCYP3A4CYP2C9PPIF
SCHEMBL19861226 0.94 PPIA (0.81) PPIAPPIBCYP3A4CYP2C9PPIF
SCHEMBL20076343 0.93 PPIA (0.70) PPIAPPIBCYP3A4CYP2C9PPIF
SCHEMBL20076105 0.92 ABCB1 (0.64) PPIAPPIBCYP3A4CYP2C9PPIF
SCHEMBL20076387 0.92 PPIA (0.75) PPIAPPIBCYP3A4CYP2C9PPIF
SCHEMBL19861299 0.91 ABCB1 (0.71) PPIAPPIBCYP3A4CYP2C9PPIF
SCHEMBL19861297 0.91 ABCB1 (0.71) PPIAPPIBCYP3A4CYP2C9PPIF
SCHEMBL19861271 0.91 PPIA (0.66) PPIAPPIBCYP3A4CYP2C9PPIF
SCHEMBL19860358 0.91 PPIA (0.68) PPIAPPIBCYP3A4CYP2C9PPIF
SCHEMBL19861197 0.91 PPIA (0.77) PPIAPPIBCYP3A4CYP2C9PPIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890198-B2 Cyclosporin derivatives and uses thereof S&T GLOBAL INC. (US) 2018-02-13 US disclosed