SCHEMBL19861629

SCHEMBL19861629

NC(=O)[C@H]1CCCN1C(=O)c1cc(NNc2cc(C(=O)N3CCSCC3)cn3nc(-c4ccco4)nc23)c2nc(-c3ccco3)nn2c1

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 15/20 0.54
ADORA3 P0DMS8 1/20 0.39
ADORA1 P30542 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18269265 0.83 ADORA2A (0.69) ADORA2A
SCHEMBL18271598 0.83 ADORA2A (0.56) ADORA2AADORA3ADORA1
SCHEMBL7043856 0.83 ADORA2A (0.69) ADORA2A
SCHEMBL6885552 0.78 ADORA2A (0.83) ADORA2A
SCHEMBL6879417 0.72 ADORA2A (0.73) ADORA2A
SCHEMBL1044059 0.71 ADORA2A (1.00) ADORA2A
SCHEMBL18271425 0.71 ADORA2A (0.59) ADORA2AADORA3ADORA1
SCHEMBL6884462 0.71 ADORA2A (1.00) ADORA2A
SCHEMBL7047131 0.69 ADORA2A (0.69) ADORA2A
SCHEMBL6879387 0.69 ADORA2A (0.73) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9889082-B2 Methods and compositions for inhibiting or reducing hair loss, acne, rosacea, prostate cancer, and BPH THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-02-13 US disclosed