Dapagliflozin

Dapagliflozin

SCHEMBL19867556

CCOc1ccc(Cc2cc(C3OC(CO)[C@@H](O)[C@H](O)[C@H]3O)ccc2Cl)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SLC5A2

The experimentally established mechanism targets of Dapagliflozin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC5A2 known ✓ P31639 20/20 1.00
SLC5A1 P13866 14/20 1.00
ADRA2A P08913 1/20 1.00
SLC5A11 Q8WWX8 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dapagliflozin SCHEMBL14949160 1.00 SLC5A2 (1.00) SLC5A2SLC5A1ADRA2ASLC5A11
Dapagliflozin SCHEMBL16155111 1.00 SLC5A2 (1.00) SLC5A2SLC5A1ADRA2ASLC5A11
Dapagliflozin SCHEMBL12781978 1.00 SLC5A2 (1.00) SLC5A2SLC5A1ADRA2ASLC5A11
Dapagliflozin SCHEMBL16001389 1.00 SLC5A2 (1.00) SLC5A2SLC5A1ADRA2ASLC5A11
Dapagliflozin SCHEMBL15906654 1.00 SLC5A2 (1.00) SLC5A2SLC5A1ADRA2ASLC5A11
Dapagliflozin SCHEMBL14149845 1.00 SLC5A2 (1.00) SLC5A2SLC5A1ADRA2ASLC5A11
Dapagliflozin SCHEMBL23542057 1.00 SLC5A2 (1.00) SLC5A2SLC5A1ADRA2ASLC5A11
Dapagliflozin SCHEMBL499725 1.00 SLC5A2 (1.00) SLC5A2SLC5A1ADRA2ASLC5A11
Dapagliflozin SCHEMBL15281296 1.00 SLC5A2 (1.00) SLC5A2SLC5A1ADRA2ASLC5A11
Dapagliflozin SCHEMBL18214900 1.00 SLC5A2 (1.00) SLC5A2SLC5A1ADRA2ASLC5A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018029611-A1 NOVEL PROCESSES FOR PREPARATION OF DAPAGLIFLOZIN OR ITS SOLVATES OR CO-CRYSTALS THEREOF LAURUS LABS LIMITED (IN) 2018-02-15 WO disclosed