SCHEMBL19869751

SCHEMBL19869751

Cc1cc(-c2ccc(CN3CCN(C)CC3)cc2)cn(C)c1=O

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 10/20 0.59
BRD9 Q9H8M2 2/20 0.59
CHKA P35790 6/20 0.56
TNKS O95271 2/20 0.50
PARP1 P09874 1/20 0.50
CHEK1 O14757 1/20 0.49
LMNA P02545 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19869833 0.90 BRD4 (0.60) BRD4BRD9CHKA
SCHEMBL19869832 0.89 BRD4 (0.59) BRD4BRD9CHKA
SCHEMBL19869742 0.87 BRD4 (0.56) BRD4BRD9TNKSCHEK1
SCHEMBL19869673 0.87 HRH3 (0.59) BRD4BRD9TNKSCHEK1
SCHEMBL19869689 0.85 BRD4 (0.51) BRD4BRD9CHKA
SCHEMBL19857636 0.82 BRD4 (0.64) BRD4BRD9
SCHEMBL19857635 0.81 BRD4 (0.47) BRD4BRD9CHKA
SCHEMBL19869701 0.80 BRD4 (0.68) BRD4BRD9
SCHEMBL19857625 0.79 BRD4 (0.50) BRD4BRD9CHKA
SCHEMBL19869706 0.79 BRD4 (0.65) BRD4BRD9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3265453-B1 NEW PYRIDINONES AND ISOQUINOLINONES AS INHIBITORS OF THE BROMODOMAIN BRD9 BOEHRINGER INGELHEIM INT (DE) 2022-06-29 EP disclosed
US-11319318-B2 Pyridinones and isoquinolinones as inhibitors of the bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-05-03 US disclosed
US-20180044335-A1 New Pyridinones and Isoquinolinones as Inhibitors of the Bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-02-15 US disclosed
US-20180044335-A1 New Pyridinones and Isoquinolinones as Inhibitors of the Bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-02-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180044335-A1 New Pyridinones and Isoquinolinones as Inhibitors of the Bromodomain BRD9 BRD9, BRD1, BRD2 BRD4 5/4885BRD9 1/4885CHKA 1326/4885
US-11319318-B2 Pyridinones and isoquinolinones as inhibitors of the bromodomain BRD9 BRD9, BRD1, BRD2 BRD4 6/4885BRD9 1/4885CHKA 1404/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.