SCHEMBL19869792

SCHEMBL19869792

COCc1c(OC)cc(-c2cc(C)c(=O)n(C)c2C)cc1OC

nearest known ligand 0.72

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRD9 Q9H8M2 16/20 0.72
BRD4 O60885 12/20 0.72
BRD7 Q9NPI1 10/20 0.72
BRD2 P25440 5/20 0.72
TAF1 P21675 1/20 0.35
TGFBR1 P36897 1/20 0.35
BRPF1 P55201 1/20 0.35
ACVR1 Q04771 1/20 0.35
BPTF Q12830 1/20 0.35
TAF1L Q8IZX4 1/20 0.35
CREBBP Q92793 1/20 0.35
CECR2 Q9BXF3 1/20 0.35
BAZ2B Q9UIF8 1/20 0.35
ATAD2B Q9ULI0 1/20 0.35
CYP19A1 P11511 3/20 0.33
NQO2 P16083 3/20 0.33
ERN1 O75460 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19869782 0.84 BRD9 (0.69) BRD9BRD4BRD7BRD2TAF1
SCHEMBL19869680 0.84 BRD9 (1.00) BRD9BRD4BRD7BRD2TAF1
SCHEMBL19869794 0.82 BRD4 (0.66) BRD9BRD4BRD7BRD2TGFBR1
SCHEMBL19869786 0.80 BRD4 (0.63) BRD9BRD4BRD7BRD2
SCHEMBL19869781 0.79 BRD4 (0.69) BRD9BRD4BRD7BRD2
SCHEMBL19869722 0.76 BRD4 (0.71) BRD9BRD4BRD7BRD2
SCHEMBL19869768 0.75 BRD9 (0.72) BRD9BRD4BRD7BRD2TAF1
SCHEMBL19869824 0.71 BRD9 (0.77) BRD9BRD4BRD7BRD2TAF1
SCHEMBL19869812 0.70 BRD4 (0.48) BRD9BRD4BRD7BRD2
SCHEMBL19869784 0.69 BRD9 (0.57) BRD9BRD4BRD7BRD2TAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3265453-B1 NEW PYRIDINONES AND ISOQUINOLINONES AS INHIBITORS OF THE BROMODOMAIN BRD9 BOEHRINGER INGELHEIM INT (DE) 2022-06-29 EP disclosed
US-11319318-B2 Pyridinones and isoquinolinones as inhibitors of the bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-05-03 US disclosed
US-20180044335-A1 New Pyridinones and Isoquinolinones as Inhibitors of the Bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-02-15 US disclosed
US-20180044335-A1 New Pyridinones and Isoquinolinones as Inhibitors of the Bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-02-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180044335-A1 New Pyridinones and Isoquinolinones as Inhibitors of the Bromodomain BRD9 BRD9, BRD1, BRD2 BRD9 1/4885BRD4 5/4885BRD7 6/4885
US-11319318-B2 Pyridinones and isoquinolinones as inhibitors of the bromodomain BRD9 BRD9, BRD1, BRD2 BRD9 1/4885BRD4 6/4885BRD7 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.