SCHEMBL19869909

SCHEMBL19869909

Cn1cc(-c2ccc(CN)cc2)c2ccccc2c1=O

nearest known ligand 0.68

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 19/20 0.68
BRD9 Q9H8M2 1/20 0.56
BRD7 Q9NPI1 1/20 0.56
BRDT Q58F21 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12205172 0.86 BRD4 (0.70) BRD4BRD9BRD7BRDT
SCHEMBL15893960 0.82 BRD4 (0.74) BRD4BRD9BRD7
SCHEMBL19869887 0.82 BRD4 (0.64) BRD4BRD9BRD7
SCHEMBL6334276 0.81 BRD4 (1.00) BRD4BRD9BRD7BRDT
SCHEMBL19857675 0.79 BRD4 (0.47) BRD4BRD9BRD7
SCHEMBL15893958 0.79 BRD4 (0.74) BRD4BRD9BRD7
SCHEMBL19869904 0.77 BRD4 (0.57) BRD4BRD9BRD7
SCHEMBL24556609 0.77 BRD4 (0.66) BRD4BRD9BRD7
SCHEMBL19869907 0.77 BRD4 (0.66) BRD4BRD9BRD7
SCHEMBL19869906 0.77 BRD4 (0.66) BRD4BRD9BRD7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3265453-B1 NEW PYRIDINONES AND ISOQUINOLINONES AS INHIBITORS OF THE BROMODOMAIN BRD9 BOEHRINGER INGELHEIM INT (DE) 2022-06-29 EP disclosed
US-11319318-B2 Pyridinones and isoquinolinones as inhibitors of the bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-05-03 US disclosed
US-20180044335-A1 New Pyridinones and Isoquinolinones as Inhibitors of the Bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-02-15 US disclosed
US-20180044335-A1 New Pyridinones and Isoquinolinones as Inhibitors of the Bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-02-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180044335-A1 New Pyridinones and Isoquinolinones as Inhibitors of the Bromodomain BRD9 BRD9, BRD1, BRD2 BRD4 5/4885BRD9 1/4885BRD7 6/4885
US-11319318-B2 Pyridinones and isoquinolinones as inhibitors of the bromodomain BRD9 BRD9, BRD1, BRD2 BRD4 6/4885BRD9 1/4885BRD7 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.