SCHEMBL19873610

SCHEMBL19873610

COc1cc(-c2sc(F)cc2NC(=O)OC(C)c2ccsc2)ccc1-c1ccc(C2CC2)cc1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.34
LPAR1 Q92633 1/20 0.34
LPAR3 Q9UBY5 1/20 0.34
NAAA Q02083 1/20 0.31
AKR1C3 P42330 1/20 0.31
AKR1C2 P52895 1/20 0.31
KDM1A O60341 1/20 0.31
MAOA P21397 1/20 0.31
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
MCHR1 Q99705 1/20 0.30
CHRM2 P08172 1/20 0.30
CHRM1 P11229 1/20 0.30
CHRM3 P20309 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
POLB P06746 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19873555 0.91 LPAR1 (0.34) APPLPAR1LPAR3NAAAAKR1C3
SCHEMBL19873553 0.91 LPAR1 (0.34) APPLPAR1LPAR3NAAAAKR1C3
SCHEMBL19873559 0.90 LPAR1 (0.37) APPLPAR1LPAR3NAAA
SCHEMBL19873600 0.90 LPAR1 (0.37) APPLPAR1LPAR3NAAA
SCHEMBL19873542 0.89 APP (0.37) APPLPAR1LPAR3NAAAAKR1C3
SCHEMBL19873541 0.89 APP (0.37) APPLPAR1LPAR3NAAAAKR1C3
SCHEMBL19873569 0.89 LPAR1 (0.43) APPLPAR1LPAR3NAAAAKR1C3
SCHEMBL19873568 0.89 LPAR1 (0.43) APPLPAR1LPAR3NAAAAKR1C3
SCHEMBL19873649 0.88 APP (0.40) APPLPAR1LPAR3NAAAAKR1C3
SCHEMBL19873572 0.88 CHRM3 (0.37) APPLPAR1LPAR3NAAAAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3360869-B1 HALOGEN-SUBSTITUTED HETEROCYCLIC COMPOUND USEFUL FOR THE TREATMENT OF DISEASES CAUSED BY LPA. UBE INDUSTRIES (JP) 2020-07-29 EP claimed
EP-2940013-B1 HALOGEN-SUBSTITUTED HETEROCYCLIC COMPOUND UBE INDUSTRIES (JP) 2018-02-21 EP claimed