SCHEMBL19873661

SCHEMBL19873661

COc1cc(-c2sc(F)cc2NC(=O)O[C@H](C)c2ccc(F)cc2Cl)ccc1-c1ccc(C2CC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 1/20 0.39
SCN9A Q15858 1/20 0.36
CHRM3 P20309 10/20 0.35
JAK2 O60674 1/20 0.34
PI4KB Q9UBF8 1/20 0.34
CHRM2 P08172 2/20 0.34
CHRM1 P11229 2/20 0.34
CTSA P10619 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19873664 1.00 LPAR1 (0.39) LPAR1SCN9ACHRM3JAK2PI4KB
SCHEMBL19873591 0.94 LPAR1 (0.40) LPAR1SCN9ACHRM3JAK2PI4KB
SCHEMBL19873589 0.94 LPAR1 (0.40) LPAR1SCN9ACHRM3JAK2PI4KB
SCHEMBL19873624 0.94 JAK2 (0.40) LPAR1CHRM3JAK2PI4KBCHRM2
SCHEMBL19873575 0.93 LPAR1 (0.43) LPAR1CHRM3
SCHEMBL19873578 0.93 LPAR1 (0.43) LPAR1CHRM3
SCHEMBL19873549 0.92 CHRM3 (0.35) LPAR1CHRM3CHRM2CHRM1CTSA
SCHEMBL19873552 0.92 CHRM3 (0.35) LPAR1CHRM3CHRM2CHRM1CTSA
SCHEMBL19873587 0.91 CHRM3 (0.34) LPAR1CHRM3CHRM2CHRM1CTSA
SCHEMBL19873627 0.91 CHRM3 (0.35) LPAR1CHRM3JAK2CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3360869-B1 HALOGEN-SUBSTITUTED HETEROCYCLIC COMPOUND USEFUL FOR THE TREATMENT OF DISEASES CAUSED BY LPA. UBE INDUSTRIES (JP) 2020-07-29 EP claimed
EP-2940013-B1 HALOGEN-SUBSTITUTED HETEROCYCLIC COMPOUND UBE INDUSTRIES (JP) 2018-02-21 EP claimed