SCHEMBL19877239

SCHEMBL19877239

[H]/N=C(/NO)c1ccc(C=Cc2c(N)ncc3ccc(Cl)cc23)cc1

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 3/20 0.40
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
KIT P10721 1/20 0.31
NTRK3 Q16288 1/20 0.31
MAP4K4 O95819 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19877236 0.92 FLT3 (0.40) FLT3KDM4ENPC1RAB9AKIT
SCHEMBL17469806 0.81 MAP4K4 (0.45) FLT3KDM4ENPC1RAB9AMAP4K4
SCHEMBL21103816 0.80 KIT (0.47) FLT3KITNTRK3
SCHEMBL19891639 0.77 FLT3 (0.35) FLT3KDM4ENPC1RAB9A
SCHEMBL19891638 0.75 FLT3 (0.44) FLT3KDM4ENPC1RAB9AMAP4K4
SCHEMBL19006326 0.74 FLT3 (0.35) FLT3KDM4ENPC1RAB9AMAP4K4
SCHEMBL21103088 0.72 HPGD (0.47) FLT3KDM4ENPC1RAB9A
SCHEMBL23573082 0.72 FLT3 (0.39) FLT3KITNTRK3MAP4K4
SCHEMBL23599921 0.70 MEN1 (0.47)
SCHEMBL19877238 0.70 FLT3 (0.68) FLT3KITNTRK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250084039-A1 4-SUBSTITUTED AMINOISOQUINOLINE DERIVATIVES PURDUE RESEARCH FOUNDATION (US) 2025-03-13 US disclosed
EP-4011882-B1 4-SUBSTITUTED AMINOISOQUINOLINE DERIVATIVES PURDUE RESEARCH FOUNDATION (US) 2025-03-05 EP disclosed
EP-4011882-A1 4-SUBSTITUTED AMINOISOQUINOLINE DERIVATIVES Purdue Research Foundation (US) 2022-06-15 EP disclosed
US-20210198208-A1 4-SUBSTITUTED AMINOISOQUINOLINE DERIVATIVES PURDUE RESEARCH FOUNDATION (US) 2021-07-01 US disclosed
US-11001559-B2 4-substituted aminoisoquinoline derivatives PURDUE RESEARCH FOUNDATION (US) 2021-05-11 US disclosed
EP-3496717-A1 4-SUBSTITUTED AMINOISOQUINOLINE DERIVATIVES Purdue Research Foundation (US) 2019-06-19 EP disclosed
US-20190177278-A1 4-SUBSTITUTED AMINOISOQUINOLINE DERIVATIVES PURDUE RESEARCH FOUNDATION (US) 2019-06-13 US disclosed
WO-2018035072-A1 4-SUBSTITUTED AMINOISOQUINOLINE DERIVATIVES PURDUE RESEARCH FOUNDATION (US) 2018-02-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190177278-A1 4-SUBSTITUTED AMINOISOQUINOLINE DERIVATIVES MCL1, ABL1, FLT3 FLT3 3/4885KDM4E 93/4885NPC1 3761/4885
US-11001559-B2 4-substituted aminoisoquinoline derivatives MCL1, ABL1, FLT3 FLT3 3/4885KDM4E 93/4885NPC1 3761/4885
US-20210198208-A1 4-SUBSTITUTED AMINOISOQUINOLINE DERIVATIVES MCL1, ABL1, FLT3 FLT3 3/4885KDM4E 93/4885NPC1 3761/4885
US-20250084039-A1 4-SUBSTITUTED AMINOISOQUINOLINE DERIVATIVES MCL1, ABL1, FLT3 FLT3 3/4885KDM4E 93/4885NPC1 3761/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.