SCHEMBL19902533

SCHEMBL19902533

CC(C)(C)OC(=O)N[C@H]1CC[C@H](c2nn(C(C3CC3)C3CC3)c(=O)c3ccccc32)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 3/20 0.45
JAK2 O60674 2/20 0.45
TYK2 P29597 1/20 0.45
JAK3 P52333 1/20 0.45
KDM1A O60341 1/20 0.42
MAOB P27338 1/20 0.42
BTK Q06187 4/20 0.41
DRD2 P14416 2/20 0.41
CHRNA7 P36544 1/20 0.40
CKS1B P61024 1/20 0.39
SKP1 P63208 1/20 0.39
SKP2 Q13309 1/20 0.39
KMT2A Q03164 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CACNB4 O00305 1/20 0.38
CACNA1A O00555 1/20 0.38
CACNA1G O43497 1/20 0.38
CACNG3 O60359 1/20 0.38
CACNA1F O60840 1/20 0.38
CACNA1H O95180 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17452549 0.89 KMT2A (0.37) JAK1JAK2TYK2JAK3KDM1A
SCHEMBL19902579 0.79 KDM1A (0.43) JAK1JAK2TYK2JAK3KDM1A
SCHEMBL19902296 0.75 JAK1 (0.49) JAK1JAK2TYK2JAK3KDM1A
SCHEMBL19902293 0.75 JAK1 (0.49) JAK1JAK2TYK2JAK3KDM1A
SCHEMBL19902295 0.75 JAK1 (0.49) JAK1JAK2TYK2JAK3KDM1A
SCHEMBL19902459 0.75 CHRNA7 (0.37) JAK1JAK2TYK2JAK3DRD2
SCHEMBL17452779 0.70 KMT2A (0.37) JAK1JAK2TYK2JAK3KDM1A
SCHEMBL19380852 0.70 KDM1A (0.68) JAK1JAK2TYK2JAK3KDM1A
SCHEMBL9638796 0.67 KDM1A (0.55) KDM1AMAOBBTKDRD2CKS1B
SCHEMBL20563839 0.67 JAK1 (0.49) JAK1JAK2TYK2JAK3KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9902702-B2 Spirocycloheptanes as inhibitors of rock BRISTOL-MYERS SQUIBB COMPANY (US) 2018-02-27 US disclosed