SCHEMBL19903083

SCHEMBL19903083

CN1Cc2cccc(C(=O)N=O)c2C1=O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.68
PARP2 Q9UGN5 5/20 0.47
HTT P42858 3/20 0.47
LMNA P02545 1/20 0.47
POLB P06746 2/20 0.41
ESR2 Q92731 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ESR1 P03372 1/20 0.41
NR4A1 P22736 1/20 0.41
APEX1 P27695 1/20 0.41
PTPN7 P35236 1/20 0.41
RECQL P46063 1/20 0.41
BLM P54132 1/20 0.41
MCL1 Q07820 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
ALOX15 P16050 1/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPK10 P53779 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL835757 0.83 PARP1 (0.74) PARP1PARP2HTTLMNAPOLB
SCHEMBL834540 0.81 PARP1 (1.00) PARP1PARP2HTTLMNAPOLB
SCHEMBL12336994 0.74 PARP1 (0.54) PARP1PARP2HTTLMNAPOLB
SCHEMBL1355339 0.74 PARP1 (0.61) PARP1PARP2HTTLMNAHSD17B10
SCHEMBL12714874 0.72 PARP1 (0.63) PARP1PARP2HTTLMNAPOLB
SCHEMBL29955619 0.71 PARP1 (0.58) PARP1PARP2HTTLMNA
SCHEMBL20468587 0.71 PARP1 (0.58) PARP1PARP2HTTLMNA
SCHEMBL14996499 0.70 PARP1 (0.57) PARP1PARP2HTTLMNA
SCHEMBL25767173 0.70 PARP1 (0.57) PARP1PARP2HTTLMNA
SCHEMBL18089021 0.70 PARP1 (0.57) PARP1PARP2HTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3287454-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2018-02-28 EP disclosed