SCHEMBL19904490

SCHEMBL19904490

CNC(=O)[C@@H]1CCN(c2ccc(Cl)cc2)C1

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 11/20 0.68
CCR1 P32246 1/20 0.49
MCHR1 Q99705 1/20 0.48
AKR1C3 P42330 1/20 0.48
SYK P43405 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
KMT2A Q03164 1/20 0.46
FFAR1 O14842 1/20 0.46
MAP4K4 O95819 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13733384 0.85 NOTUM (0.57) NOTUMSYKMAPK1MAP4K4
SCHEMBL21339818 0.82 NOTUM (0.68) NOTUMAKR1C3MEN1ALDH1A1LMNA
SCHEMBL3440331 0.82 NOTUM (0.54) NOTUMSYKMAP4K4
SCHEMBL20840870 0.82 NOTUM (0.68) NOTUMAKR1C3MEN1ALDH1A1LMNA
SCHEMBL16695183 0.81 NOTUM (1.00) NOTUMAKR1C3FFAR1
SCHEMBL895254 0.81 NOTUM (1.00) NOTUMAKR1C3FFAR1
SCHEMBL16695070 0.80 NOTUM (0.74) NOTUMAKR1C3HDAC1HDAC8HDAC6
SCHEMBL16695071 0.80 NOTUM (0.74) NOTUMAKR1C3HDAC1HDAC8HDAC6
SCHEMBL16695087 0.80 NOTUM (0.74) NOTUMAKR1C3HDAC1HDAC8HDAC6
SCHEMBL16994779 0.78 TSHR (0.53) NOTUMSYKMEN1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3063141-B1 N-(1-HYDROXY-3-(PYRROLIDINYL)PROPAN-2-YL)PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS BIOMARIN PHARM INC (US) 2018-02-28 EP disclosed