SCHEMBL19905065

SCHEMBL19905065

CN1CCOc2cc(-c3cc(N)ncn3)ccc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.52
CYP11B2 P19099 1/20 0.52
NOTUM Q6P988 1/20 0.49
KMO O15229 1/20 0.43
HDAC4 P56524 1/20 0.43
KDM5B Q9UGL1 1/20 0.42
ASIC3 Q9UHC3 1/20 0.41
GRM5 P41594 1/20 0.40
METAP2 P50579 1/20 0.39
LCK P06239 1/20 0.39
TNK2 Q07912 1/20 0.39
EIF2AK3 Q9NZJ5 1/20 0.39
MET P08581 1/20 0.39
PIK3CA P42336 2/20 0.38
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
RECQL P46063 1/20 0.37
PTGES2 Q9H7Z7 1/20 0.37
POLQ O75417 1/20 0.37
PIK3CD O00329 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15345147 0.79 CYP11B1 (0.57) CYP11B1CYP11B2NOTUMHDAC4KDM5B
SCHEMBL15473162 0.77 PIK3CA (0.45) CYP11B1CYP11B2NOTUMKDM5BLCK
SCHEMBL15341897 0.75 CYP11B1 (0.53) CYP11B1CYP11B2NOTUMHDAC4KDM5B
SCHEMBL14320634 0.73 CYP11B1 (0.64) CYP11B1CYP11B2NOTUMHDAC4KDM5B
SCHEMBL3582361 0.73 CYP11B1 (0.51) CYP11B1CYP11B2NOTUMHDAC4ALDH1A1
SCHEMBL10187283 0.72 ADORA2A (0.57) KMOASIC3LCKTNK2MET
SCHEMBL15345191 0.69 CCR1 (0.47) CYP11B1CYP11B2NOTUMGRM5METAP2
SCHEMBL154510 0.68 CYP11B1 (0.52) CYP11B1CYP11B2NOTUMHDAC4PIK3CA
SCHEMBL2334976 0.68 CYP11B1 (0.52) CYP11B1CYP11B2NOTUMHDAC4KDM5B
SCHEMBL25094648 0.68 CYP11B1 (0.53) CYP11B1CYP11B2NOTUMHDAC4KDM5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057959-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2018-02-28 EP disclosed