SCHEMBL19905253

SCHEMBL19905253

CNC(=O)c1c(F)cnc2c(C(C)CNc3cc(-c4cnc(NCC(F)(F)F)nc4)ncn3)cccc12

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 2/20 0.44
FAAH O00519 16/20 0.36
ABL1 P00519 1/20 0.34
BCR P11274 1/20 0.34
KDR P35968 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17874697 1.00 PRKDC (0.44) PRKDCFAAHABL1BCRKDR
SCHEMBL17634922 0.92 PRKDC (0.46) PRKDCFAAHABL1BCR
SCHEMBL17874736 0.90 PRKDC (0.45) PRKDCFAAHABL1BCR
SCHEMBL15339625 0.89 PRKDC (0.55) PRKDCFAAHABL1BCR
SCHEMBL15339667 0.89 PRKDC (0.48) PRKDCFAAHABL1BCR
SCHEMBL17874692 0.89 PRKDC (0.46) PRKDCFAAH
SCHEMBL15473127 0.88 PRKDC (0.43) PRKDCFAAHABL1BCR
SCHEMBL17874737 0.88 PRKDC (0.45) PRKDCFAAH
SCHEMBL17874718 0.88 PRKDC (0.43) PRKDCFAAHABL1BCR
SCHEMBL16665021 0.88 PRKDC (0.45) PRKDCFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057959-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2018-02-28 EP disclosed