SCHEMBL19905286

SCHEMBL19905286

CNC(=O)c1ccnc2c(C(C)CCNc3cc(-c4ccc(OC(C)(C)C)cc4)ncn3)cccc12

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 7/20 0.39
BCR P11274 6/20 0.39
PRKDC P78527 2/20 0.39
FAAH O00519 5/20 0.37
SLC40A1 Q9NP59 1/20 0.35
LRRK2 Q5S007 1/20 0.35
USP2 O75604 3/20 0.35
CYP1A2 P05177 3/20 0.35
CYP3A4 P08684 3/20 0.35
CYP2C19 P33261 3/20 0.35
CLK4 Q9HAZ1 3/20 0.35
ALDH1A1 P00352 2/20 0.34
CYP2D6 P10635 2/20 0.34
ALOX15 P16050 2/20 0.34
MEN1 O00255 1/20 0.34
CYP2C9 P11712 1/20 0.34
KMT2A Q03164 1/20 0.34
PIK3CA P42336 1/20 0.34
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17634758 0.92 PRKDC (0.46) ABL1BCRPRKDCFAAHSLC40A1
SCHEMBL19355283 0.88 PRKDC (0.41) ABL1BCRPRKDCFAAHSLC40A1
SCHEMBL20373542 0.87 PRKDC (0.40) ABL1BCRPRKDCFAAHSLC40A1
SCHEMBL19355572 0.87 PRKDC (0.40) ABL1BCRPRKDCFAAHSLC40A1
SCHEMBL20373149 0.86 PRKDC (0.38) ABL1BCRPRKDCFAAHSLC40A1
SCHEMBL19355279 0.86 PRKDC (0.43) ABL1BCRPRKDCFAAHSLC40A1
SCHEMBL20373549 0.86 PRKDC (0.44) ABL1BCRPRKDCFAAHSLC40A1
SCHEMBL19355288 0.86 CYP1A2 (0.43) ABL1BCRFAAHSLC40A1USP2
SCHEMBL20373509 0.86 PRKDC (0.45) PRKDCFAAHSLC40A1LRRK2USP2
SCHEMBL19355516 0.85 PRKDC (0.39) PRKDCFAAHSLC40A1LRRK2USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057959-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2018-02-28 EP disclosed