SCHEMBL19906033

SCHEMBL19906033

Cc1ccc(-c2c(CC(=O)O)c(C)cc3nc(-c4cc(-c5ccc6c(cnn6C)c5)ccn4)sc23)cc1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.37
GFER P55789 2/20 0.37
POLQ O75417 1/20 0.36
CACNA1H O95180 1/20 0.35
USP7 Q93009 1/20 0.35
CCNC P24863 3/20 0.34
CDK8 P49336 3/20 0.34
KMT2A Q03164 1/20 0.33
NOTUM Q6P988 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TGFBR1 P36897 1/20 0.32
MAPK14 Q16539 1/20 0.32
AR P10275 4/20 0.31
WNT1 P04628 1/20 0.31
CLK2 P49760 1/20 0.31
CLK3 P49761 1/20 0.31
GSK3B P49841 1/20 0.31
DYRK1A Q13627 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906378 0.94 PTGDR2 (0.35) KDM4EGFERPOLQCACNA1HUSP7
SCHEMBL19905859 0.89 PTGDR2 (0.37) KDM4EPOLQCACNA1HUSP7CCNC
SCHEMBL19906374 0.84 POLQ (0.33) KDM4EPOLQUSP7CCNCCDK8
SCHEMBL19906023 0.84 PTGDR2 (0.35) KDM4EPOLQKMT2AALDH1A1
SCHEMBL17547145 0.84 PTGDR2 (0.35) KDM4EPOLQCACNA1HUSP7CCNC
SCHEMBL19906180 0.84 PTGDR2 (0.41) KDM4EPOLQCACNA1HUSP7CCNC
SCHEMBL19906048 0.83 PTGDR2 (0.38) KDM4EPOLQUSP7KMT2AALDH1A1
SCHEMBL19906009 0.83 PTGDR2 (0.35) KDM4EPOLQUSP7CCNCCDK8
SCHEMBL17547144 0.83 PTGDR2 (0.35) KDM4EKMT2AALDH1A1
SCHEMBL19906010 0.83 KDM4E (0.36) KDM4EPOLQUSP7KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed