SCHEMBL19906165

SCHEMBL19906165

Cc1cc2nc(-c3ccc4c(c3)c(=O)n(C)n4C)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.40
PTGDR2 Q9Y5Y4 8/20 0.39
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
AKR1B1 P15121 1/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
HPGD P15428 1/20 0.35
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
MCHR1 Q99705 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 1/20 0.34
POLB P06746 1/20 0.34
RAB9A P51151 1/20 0.34
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
PDE5A O76074 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905816 0.93 KDM4E (0.35) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906171 0.87 KDM4E (0.36) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19905985 0.86 KDM4E (0.35) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19905960 0.86 KDM4E (0.42) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19905890 0.85 PTGDR2 (0.42) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19905855 0.84 KDM4E (0.39) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906198 0.83 NPC1 (0.40) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19905953 0.83 KDM4E (0.42) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906180 0.83 PTGDR2 (0.41) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906074 0.83 KDM4E (0.38) KDM4EPTGDR2ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed