SCHEMBL19906212

SCHEMBL19906212

Cc1cc2nc(-c3ccc4c(N(C)C)nn(C)c4c3)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.38
PTGDR2 Q9Y5Y4 10/20 0.37
ALDH1A1 P00352 3/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
PDE5A O76074 1/20 0.35
PDE1A P54750 1/20 0.35
PDE1B Q01064 1/20 0.35
PDE4D Q08499 1/20 0.35
PDE7A Q13946 1/20 0.35
PDE1C Q14123 1/20 0.35
PDE3A Q14432 1/20 0.35
MAT2A P31153 2/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33
STAT6 P42226 1/20 0.32
HIF1A Q16665 1/20 0.32
AKR1B1 P15121 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906074 0.93 KDM4E (0.38) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906186 0.90 KDM4E (0.42) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906286 0.87 KDM4E (0.38) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19905960 0.84 KDM4E (0.42) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906245 0.84 HDAC3 (0.37) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19905855 0.83 KDM4E (0.39) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906248 0.83 CNR1 (0.35) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19905978 0.83 PTGDR2 (0.40) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19905953 0.82 KDM4E (0.42) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906148 0.82 PTGDR2 (0.39) KDM4EPTGDR2ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed