SCHEMBL19906233

SCHEMBL19906233

Cc1cc2nc(-c3ccnc(-c4cnc5ncn(C)c5c4)c3)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 10/20 0.34
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
KDM4C Q9H3R0 2/20 0.34
KDM5B Q9UGL1 2/20 0.34
KDM5A P29375 1/20 0.34
CYP2C19 P33261 2/20 0.31
PTGS1 P23219 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31
PTGDR Q13258 1/20 0.31
MAP4K4 O95819 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905939 0.89 PTGDR2 (0.35) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906231 0.88 KDM4C (0.33) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906317 0.87 PTGDR2 (0.35) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906402 0.86 PTGDR2 (0.36) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19905872 0.85 PTGDR2 (0.37) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL17547144 0.85 PTGDR2 (0.35) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19905852 0.85 KDM4E (0.35) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906198 0.85 NPC1 (0.40) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19905859 0.85 PTGDR2 (0.37) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19905804 0.84 PTGDR2 (0.38) PTGDR2KDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed