SCHEMBL19922282

SCHEMBL19922282

COCCN1CCN(c2cc3c(Nc4ccc(C)cc4F)c(C(N)=O)nnc3cc2OC)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 1.00
SCN5A Q14524 12/20 1.00
CSF1R P07333 6/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1276898 0.93 SCN5A (1.00) KCNH2SCN5ACSF1R
SCHEMBL29684537 0.93 SCN5A (1.00) KCNH2SCN5ACSF1R
SCHEMBL1276807 0.90 SCN5A (1.00) KCNH2SCN5ACSF1R
SCHEMBL1580922 0.90 KCNH2 (1.00) KCNH2SCN5ACSF1R
SCHEMBL1579605 0.90 SCN5A (0.83) KCNH2SCN5ACSF1R
SCHEMBL1579915 0.87 SCN5A (0.81) KCNH2SCN5ACSF1R
SCHEMBL1579528 0.87 KCNH2 (0.77) KCNH2SCN5ACSF1R
SCHEMBL1579537 0.87 SCN5A (0.81) KCNH2SCN5ACSF1R
SCHEMBL1579655 0.87 SCN5A (0.81) KCNH2SCN5ACSF1R
SCHEMBL1579889 0.86 SCN5A (0.83) KCNH2SCN5ACSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180068053-A1 SYSTEMS AND METHODS OF SELECTING COMPOUNDS WITH REDUCED RISK OF CARDIOTOXICITY USING CARDIAC SODIUM ION CHANNEL MODELS UNIV ALBERTA (CA) 2018-03-08 US disclosed
US-20180068053-A1 SYSTEMS AND METHODS OF SELECTING COMPOUNDS WITH REDUCED RISK OF CARDIOTOXICITY USING CARDIAC SODIUM ION CHANNEL MODELS UNIV ALBERTA (CA) 2018-03-08 US disclosed
US-20180068053-A1 SYSTEMS AND METHODS OF SELECTING COMPOUNDS WITH REDUCED RISK OF CARDIOTOXICITY USING CARDIAC SODIUM ION CHANNEL MODELS UNIV ALBERTA (CA) 2018-03-08 US disclosed