SCHEMBL19930726

SCHEMBL19930726

CSc1ccc(OCC2CC2)c(-c2cn(C)c(=O)c3ccc(F)cc23)n1

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 19/20 0.52
KDM5A P29375 1/20 0.40
KDM4C Q9H3R0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19930681 0.97 BRD4 (0.52) BRD4KDM5AKDM4C
SCHEMBL29849058 0.84 BRD4 (0.51) BRD4
SCHEMBL16652199 0.84 BRD4 (0.51) BRD4
SCHEMBL25043103 0.84 BRD4 (0.54) BRD4KDM5AKDM4C
SCHEMBL21916735 0.84 BRD4 (0.50) BRD4KDM5AKDM4C
SCHEMBL19930659 0.82 BRD4 (0.50) BRD4KDM5AKDM4C
SCHEMBL19931478 0.82 BRD4 (0.47) BRD4KDM5AKDM4C
SCHEMBL29848254 0.81 BRD4 (0.52) BRD4
SCHEMBL16650319 0.81 BRD4 (0.52) BRD4
SCHEMBL25043223 0.80 BRD4 (0.40) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4134364-A2 BROMODOMAIN INHIBITORS Celgene Quanticel Research, Inc. (US) 2023-02-15 EP disclosed
EP-3640241-A1 BROMODOMAIN INHIBITORS Celgene Quanticel Research, Inc. (US) 2020-04-22 EP disclosed
EP-3290407-A1 BROMODOMAIN INHIBITORS Celgene Quanticel Research, Inc (US) 2018-03-07 EP disclosed