SCHEMBL19937997

SCHEMBL19937997

N#Cc1cc(-c2ccn(CC3CC3)n2)cnc1N

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 8/20 0.52
MAP3K14 Q99558 1/20 0.40
PKM P14618 1/20 0.36
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
CDC42BPB Q9Y5S2 1/20 0.36
PIK3CA P42336 1/20 0.35
FGFR1 P11362 1/20 0.35
FGFR2 P21802 1/20 0.35
FGFR3 P22607 1/20 0.35
XDH P47989 1/20 0.35
RORC P51449 1/20 0.35
TNIK Q9UKE5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19937617 0.81 MAP3K12 (0.50) MAP3K12FGFR1FGFR2FGFR3
SCHEMBL19937851 0.81 MAP3K12 (0.51) MAP3K12PIK3CAFGFR1FGFR2FGFR3
SCHEMBL19937665 0.79 MAP3K12 (0.52) MAP3K12
SCHEMBL19937780 0.79 MAP3K12 (0.52) MAP3K12FGFR1FGFR2FGFR3
SCHEMBL19938095 0.77 MAP3K12 (0.52) MAP3K12ROCK2ROCK1CDC42BPBPIK3CA
SCHEMBL19937864 0.76 MAP3K12 (0.52) MAP3K12FGFR1FGFR2FGFR3
SCHEMBL19937750 0.76 MAP3K12 (0.55) MAP3K12
SCHEMBL19937631 0.74 MAP3K12 (0.54) MAP3K12
SCHEMBL2579099 0.74 CREBBP (0.45)
SCHEMBL19937621 0.73 MAP3K12 (0.47) MAP3K12MAP3K14ROCK2ROCK1CDC42BPB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2945938-B1 3-SUBSTITUTED PYRAZOLES AND USE AS DLK INHIBITORS HOFFMANN LA ROCHE (CH) 2018-03-07 EP disclosed