SCHEMBL19953065

SCHEMBL19953065

Fc1cccc(F)c1-c1cncn1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 9/20 0.46
IDO1 P14902 8/20 0.46
HSP90AA1 P07900 4/20 0.43
HSP90AB1 P08238 4/20 0.43
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
SRC P12931 1/20 0.36
FGFR1 P11362 1/20 0.36
MAPK14 Q16539 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1076208 0.85 HSP90AA1 (0.45) TDO2IDO1HSP90AA1HSP90AB1CYP11B1
SCHEMBL19953054 0.81 IDO1 (0.39) TDO2IDO1HSP90AA1HSP90AB1
SCHEMBL19967304 0.78 HSP90AA1 (0.49) TDO2IDO1HSP90AA1HSP90AB1
SCHEMBL12676747 0.76 CYP11B1 (0.50) IDO1HSP90AA1HSP90AB1CYP11B1CYP11B2
SCHEMBL1133124 0.73 HSP90AA1 (0.41) TDO2IDO1HSP90AA1HSP90AB1CYP11B1
SCHEMBL27989475 0.72 HTT (0.45) TDO2IDO1HSP90AA1HSP90AB1CYP11B1
SCHEMBL19953047 0.72 HSP90AA1 (0.45) HSP90AA1HSP90AB1CYP11B1CYP11B2
SCHEMBL19953169 0.72 CYP3A4 (0.43) TDO2IDO1
SCHEMBL19953094 0.71 HSP90AA1 (0.44) HSP90AA1HSP90AB1CYP11B1CYP11B2
SCHEMBL1075925 0.71 HSP90AA1 (0.47) HSP90AA1HSP90AB1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018048969-A1 MULTI-TARGETED HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-03-15 WO disclosed